{"id":5154,"date":"2024-01-16T12:26:29","date_gmt":"2024-01-16T12:26:29","guid":{"rendered":"https:\/\/farlong.com\/?p=5154"},"modified":"2024-01-27T10:27:40","modified_gmt":"2024-01-27T10:27:40","slug":"breviscapine-a-review-on-its-phytochemistry-pharmacokinetics-and-therapeutic-effects","status":"publish","type":"post","link":"https:\/\/directcm.com\/ko\/breviscapine-a-review-on-its-phytochemistry-pharmacokinetics-and-therapeutic-effects\/","title":{"rendered":"\ube0c\ub808\ube44\uc2a4\uce74\ud540: \uc2dd\ubb3c\ud654\ud559, \uc57d\ub3d9\ud559 \ubc0f \uce58\ub8cc \ud6a8\uacfc\uc5d0 \ub300\ud55c \uac80\ud1a0"},"content":{"rendered":"<div class=\"inline-authors\">\n<div class=\"authors\">\n<div class=\"authors-list\"><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Wen+L&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Luan Wen\">Luan Wen<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=He+T&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Ting He\">Ting He<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Yu+A&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"AXiang Yu\">AXiang Yu<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Sun+S&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Siqi Sun\">Siqi Sun<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Li+X&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Xiang Li\">Xiang Li<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Wei+J&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Jing Wei\">Jing Wei<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Song+R&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Ruolan Song\">Ruolan Song<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Yan+X&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Xin Yan\">Xin Yan<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Li+R&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Ruiwen Li\">Ruiwen Li<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Ren+X&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Xueyang Ren\">Xueyang Ren<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Wang+Y&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Yu Wang\">Yu Wang<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Liu+X&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Xiaoyun Liu\">Xiaoyun Liu<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Dong+Y&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Ying Dong\">Ying Dong<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Fu+X&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Xueyan Fu\">Xueyan Fu<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Pharmacy, Ningxia Medical University, Ningxia 750004, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-2\">2<\/a><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"Key Laboratory of Hui Ethnic Medicine Modernization, Ministry of Education, Ningxia 750004, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-3\">3<\/a><\/sup><span class=\"comma\">,\u00a0<\/span><\/span><span class=\"authors-list-item \"><a class=\"full-name\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=She+G&amp;cauthor_id=34263720\" data-ga-category=\"search\" data-ga-action=\"author_link\" data-ga-label=\"Gaimei She\">Gaimei She<\/a><sup class=\"affiliation-links\"><span class=\"author-sup-separator\">\u00a0<\/span><a class=\"affiliation-link\" title=\"School of Chinese Materia Medica, Beijing University of Chinese Medicine, Beijing 102488, P. R. China.\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/34263720\/#full-view-affiliation-1\">1<\/a><\/sup><\/span><\/div>\n<div><\/div>\n<\/div>\n<\/div>\n<ul id=\"full-view-identifiers\" class=\"identifiers\">\n<li><span class=\"identifier pubmed\"><span class=\"id-label\">PMID:\u00a0<\/span><strong class=\"current-id\" title=\"PubMed ID\">34263720<\/strong><\/span><\/li>\n<li><span class=\"identifier doi\"><span class=\"id-label\">DOI:\u00a0<\/span><a class=\"id-link\" href=\"https:\/\/doi.org\/10.1142\/s0192415x21500646\" target=\"_blank\" rel=\"noopener\" data-ga-category=\"full_text\" data-ga-action=\"DOI\">10.1142\/S0192415X21500646<\/a><\/span><\/li>\n<\/ul>\n<div id=\"abstract\" class=\"abstract\">\n<h2 class=\"title\">Abstract<\/h2>\n<div id=\"eng-abstract\" class=\"abstract-content selected\">\n<p>Breviscapine is one of the extracts of several flavonoids of\u00a0<i>Erigeron breviscapus<\/i>. Scutellarin is the main active component of breviscapine, and the qualitative or quantitative criteria as well. Scutellarin and its analogs share a similar skeleton of the flavonoids. Breviscapine has been widely used in the treatment of cerebral infarction and its sequelae, cerebral thrombus, coronary heart disease (CHD), and angina pectoris. Breviscapine has a broad spectrum of pharmacological activities, such as increasing blood flow, improving microcirculation, dilating blood vessels, decreasing blood viscosity, promoting fibrinolysis, inhibiting platelet aggregation, and thrombosis formation, etc. In addition, breviscapine and its analogs have significant value for drug research and development because of the superiority of those significant bioactivities. Furthermore, an increasing number of pharmacokinetic studies have explored the mechanism of scutellarin and its analogs. To provide a comprehensive understanding of the current research on breviscapine, scutellarin, and the analogs, the structural features, distribution situation, preparation method, content determination method, clinical applications, pharmacological action as well as pharmacokinetics are summarized in the present review.<\/p>\n<\/div>\n<p><strong class=\"sub-title\">Keywords:\u00a0<\/strong>Breviscapine; Pharmacokinetics; Pharmacology; Review; Scutellarin.<\/p>\n<\/div>\n<p id=\"disclaimer\" class=\"disclaimer\"><a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/disclaimer\/\" target=\"_blank\" rel=\"noopener\">PubMed Disclaimer<\/a><\/p>\n<div id=\"similar\" class=\"similar-articles\">\n<div id=\"similar\" class=\"similar-articles\">\n<h2 class=\"title\">Similar articles<\/h2>\n<ul id=\"similar-articles-list\" class=\"articles-list\">\n<li class=\"full-docsum\">\n<div class=\"docsum-content\"><a class=\"docsum-title\" href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/17354170\/\" data-ga-category=\"similar_article\" data-ga-action=\"17354170\" data-ga-label=\"\">Two major urinary metabolites of scutellarin in rats.<\/a><\/p>\n<div class=\"docsum-citation full-citation\"><span class=\"docsum-authors full-authors\">Qiu F, Xia H, Zhang T, Di X, Qu G, Yao X.<\/span><span class=\"docsum-journal-citation full-journal-citation\">Planta Med. 2007 Apr;73(4):363-5. doi: 10.1055\/s-2007-967128. 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Scutellarin is the main active component of breviscapine, and the qualitative or quantitative criteria as well. Scutellarin and its analogs share a similar skeleton of the flavonoids. Breviscapine has been widely used in the treatment of cerebral infarction and its sequelae, cerebral thrombus, coronary heart disease (CHD), and angina pectoris. <\/p>","protected":false},"author":1,"featured_media":5368,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"site-sidebar-layout":"default","site-content-layout":"","ast-site-content-layout":"default","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","theme-transparent-header-meta":"default","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"set","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"var(--ast-global-color-4)","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-gradient":""},"tablet":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-gradient":""},"mobile":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-gradient":""}},"ast-content-background-meta":{"desktop":{"background-color":"var(--ast-global-color-5)","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-gradient":""},"tablet":{"background-color":"var(--ast-global-color-5)","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-gradient":""},"mobile":{"background-color":"var(--ast-global-color-5)","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-gradient":""}},"footnotes":""},"categories":[9],"tags":[],"class_list":["post-5154","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-supplements"],"_links":{"self":[{"href":"https:\/\/directcm.com\/ko\/wp-json\/wp\/v2\/posts\/5154","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/directcm.com\/ko\/wp-json\/wp\/v2\/posts"}],"about":[{"href":"https:\/\/directcm.com\/ko\/wp-json\/wp\/v2\/types\/post"}],"author":[{"embeddable":true,"href":"https:\/\/directcm.com\/ko\/wp-json\/wp\/v2\/users\/1"}],"replies":[{"embeddable":true,"href":"https:\/\/directcm.com\/ko\/wp-json\/wp\/v2\/comments?post=5154"}],"version-history":[{"count":0,"href":"https:\/\/directcm.com\/ko\/wp-json\/wp\/v2\/posts\/5154\/revisions"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/directcm.com\/ko\/wp-json\/wp\/v2\/media\/5368"}],"wp:attachment":[{"href":"https:\/\/directcm.com\/ko\/wp-json\/wp\/v2\/media?parent=5154"}],"wp:term":[{"taxonomy":"category","embeddable":true,"href":"https:\/\/directcm.com\/ko\/wp-json\/wp\/v2\/categories?post=5154"},{"taxonomy":"post_tag","embeddable":true,"href":"https:\/\/directcm.com\/ko\/wp-json\/wp\/v2\/tags?post=5154"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}